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CB1 antagonist 5

CAT: 0804-HY-120653-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-120653-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CB1 antagonist 5 (Compound 25) is an antagonist for CB1 cannabinoid receptor, with a Ki of 243 nM and an EC50 of 195 nM[1].
CAS Number
878533-35-8
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cb1-antagonist-5.html
Smiles
O=C1N(C(C(N1C2=CC=C(C=C2)Br)C3=CC=CC=C3)=O)C4=CC=C(C=C4)Br
Molecular Formula
C21H14Br2N2O2
Molecular Weight
486.16
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
References & Citations
[1]Muccioli GG, et al., Synthesis and activity of 1,3,5-triphenylimidazolidine-2,4-diones and 1,3,5-triphenyl-2-thioxoimidazolidin-4-ones: characterization of new CB1 cannabinoid receptor inverse agonists/antagonists. J Med Chem. 2006 Feb 9;49 (3) :872-82.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB1

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