[Dmt1]DALDA

• Description:

  [Dmt1]DALDA is a potent and long-acting analgesic binds to the mu opioid receptor with high affinity and selectivity. [Dmt1]DALDA is a full agonist at hMOR (Kd = 0.199 nM) and hDOR, but only partial agonist against hKOR[1][2].

• UNSPSC:

  12352209

• Target:

  Opioid Receptor

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Others

• Smiles:

  CC (C=C (C=C1C) O) =C1C[C@H] (N) C (N[C@H] (CCCNC (N) =N) C (N[C@H] (C (N[C@H] (C (N) =O) CCCCN) =O) CC2=CC=CC=C2) =O) =O

• Molecular Formula:

  C32H49N9O5

• Molecular Weight:

  639.79

• References & Citations:

  [1]Zhao, G. M., et al., (2003) . Comparison of [Dmt1]DALDA and DAMGO in binding and G protein activation at mu, delta, and kappa opioid receptors. The Journal of pharmacology and experimental therapeutics, 307 (3), 947–954.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Peptides

• Clinical Information:

  No Development Reported

• CAS Number:

  255861-98-4