AP-503

• Description:

  AP-503 is a selective GPR133/ADGRD1 agonist with an EC50 of 1.21 nM. AP-503 is used in research on the prevention of muscle-related diseases and vestibular dysfunction[1].

• UNSPSC:

  12352005

• Target:

  Adhesion G Protein-coupled Receptors (AGPCRs)

• Related Pathways:

  GPCR/G Protein

• Field of Research:

  Others

• Purity:

  99.84

• Solubility:

  DMSO : 25 mg/mL (ultrasonic; warming; heat to 60°C)

• Smiles:

  CCN1CCN(C2=CC=C(C(OC)=O)C=C2NC(COC(C(C)=C3)=CC=C3C)=O)CC1

• Molecular Formula:

  C24H31N3O4

• Molecular Weight:

  425.52

• References & Citations:

  [1]Sun jin peng, et al. G protein coupled receptor GPR133/ADGRD1 agonist, preparation method and application thereof. CN118146176B.2024-11-15.

• Shipping Conditions:

  Blue Ice

• Storage Conditions:

  -20°C, 3 years (Powder)

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  [767299-99-0]