BP 2-94

• Description :

  BP 2-94 (BP 2.94) is an orally active and highly selective prodrug targeting the histamine H3 receptor. BP 2-94 exerts anti-inflammatory, analgesic and antinociceptive effects by inhibiting histamine release and modulating neurogenic inflammation. BP 2-94 is promising for research of asthma, migraines, and inflammatory pain-related disorders[1].

• CAS Number :

  [139191-80-3]

• Product Name Alternative :

  BP 2.94

• UNSPSC :

  12352005

• Target :

  Histamine Receptor

• Related Pathways :

  GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

• Field of Research :

  Neurological Disease

• Smiles :

  OC1=C(C=CC=C1)/C(C2=CC=CC=C2)=N\[C@@H](CC3=CN=CN3)C

• Molecular Formula :

  C19H19N3O

• Molecular Weight :

  305.37

• References & Citations :

  [1]Rouleau A, et al. Bioavailability, antinociceptive and antiinflammatory properties of BP 2-94, a histamine H3 receptor agonist prodrug. J Pharmacol Exp Ther. 1997 Jun;281 (3) :1085-94.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  H3 Receptor