Products for Research Use Only
RegisterLogin

PF-03246799 (monohydrochloride)

CAT: 0804-HY-119103BSize: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-119103BSize:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
PF-03246799 monohydrochloride is a potent and selective 5-HT2C receptor agonist with an EC50 of 190 nM and a Ki of 160 nM. PF-03246799 monohydrochloride shows selectivity for 5-HT2C over 5-HT2A and 5-HT2B receptors. PF-03246799 monohydrochloride has the potential for stress urinary incontinence (SUI) research[1].
CAS Number
1613666-08-2
UNSPSC
12352005
Target
5-HT Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Smiles
C12=NC(CC3=CC=CC=C3)=NC=C1CCNCC2.Cl
Molecular Formula
C15H18ClN3
Molecular Weight
275.78
References & Citations
[1]Andrews MD, et al. Pyrimido[4,5-d]azepines as potent and selective 5-HT2C receptor agonists: design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence. Bioorg Med Chem Lett. 2011 May 1;21 (9) :2715-20.
Shipping Conditions
Room temperature
Scientific Category
Reference compound
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor

Related Products

CatalogName
HY-119103PF-03246799
HY-W614725-01Apcin-A (monohydrochloride)
HY-15260A-01XL413 (monohydrochloride)
HY-B0502A-01Enrofloxacin (monohydrochloride)
HY-111388A-01Romaciclib (monohydrochloride)
HY-129841-01Niguldipine (monohydrochloride)
HY-50767A-01Palbociclib (monohydrochloride)
HY-B2209A-01Hydroxocobalamin (monohydrochloride)
HY-14551COsanetant (monohydrochloride)
HY-B0356A-01Ciprofloxacin (monohydrochloride)

Alternative Products

CatalogName
M10282-01PF-03246799
GTR19209166-01PF-03246799 hydrochloride
FG183203-01GSK3008348 monohydrochloride
T0250-01Ciprofloxacin monohydrochloride
T71358-01Nialamide monohydrochloride
442587-01BEPP Monohydrochloride
MBS3845814-01Foliglurax monohydrochloride
JH89478LGH447 monohydrochloride
GE9458-25gAdenine monohydrochloride
abx184117-01Hydrazine monohydrochloride

Popular Products