MOR agonist-4

• Target:

  Opioid Receptor

• Related Pathways:

  Endocrinology/Hormones|||Neuroscience|||GPCR/G Protein

• Bioactivity:

  MOR agonist-4 (2d), having an EC50 of 11 nM, is a G protein-biased agonist of the Kappa opioid receptor (KOR) . This compound features a triazole-based, electron-withdrawing CF3 group and a bias factor of 38. MOR agonist-4 is utilized for antipruritic and analgesic applications.

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C