Veldoreotide TFA

CAT: 0931-MF-0120012-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0120012-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2126831-23-8
Target
Somatostatin|||Others
Related Pathways
GPCR/G Protein|||Others
Bioactivity
Veldoreotide (DG3173) TFA, a somatostatin analogue, effectively binds to and activates somatostatin receptors (SSTR) 2, 4, and 5. This compound demonstrates a higher efficacy in inhibiting growth hormone (GH) secretion in adenomas than Octreotide, showcasing its potential as a pain modulating agent [1].
Smiles
C(C(O)=O)(F)(F)F.C(C=1C=2C(NC1)=CC=CC2)[C@H]3C(=O)N[C@H](CC=4C=5C(NC4)=CC=CC5)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]([C@@H](C)O)(C(=O)N[C@@H](CC6=CC=CC=C6)C(=O)N(CC(N)=O)CCCC(=O)NCCCC(=O)N[C@@H](CC7=CC=CC=C7)C(=O)N3)[H]
Molecular Formula
C62H75F3N12O12
Molecular Weight
1237.33
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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