BIM-23027

• Target :

  Dopamine Receptor|||Somatostatin

• Related Pathways :

  GPCR/G Protein|||Neuroscience

• Bioactivity :

  BIM-23027 is a selective sst 2 receptor agonist (EC 50 = 0.32 nM) with effects analogous to the cyclic tetradecapeptide somatostatin (SRIF) . It promotes dopamine release through a Glu-dependent mechanism [1] [2].

• Smiles :

  C(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](C)N(C)C(=O)[C@H](CC5=CC=CC=C5)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@H](CCCCN)NC3=O)[H]

• Molecular Formula :

  C43H54N8O7

• Molecular Weight :

  794.94

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  78981-49-4