LU-002i

• Target:

  Proteasome

• Related Pathways:

  Ubiquitination|||Proteases/Proteasome

• Bioactivity:

  LU-002i is a selective inhibitor targeting the human proteasome subunits ?2c and ?2i, demonstrating an inhibitory concentration (IC50) of 220 nM for ?2i [1].

• Smiles:

  C([C@@H](C(=O)[C@@]1(C)CO1)NC([C@H](CC2=CC=C(OC)C=C2)NC([C@@H](NC(CN3CCOCC3)=O)C)=O)=O)C4C5(C(CCC4)(CCCC5)[H])[H]

• Molecular Formula:

  C35H52N4O7

• Molecular Weight:

  640.81

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1838705-22-8