PHD-IN-1

CAT: 0931-T79797-01Size: 5 mgDry Ice: NoHazardous: No

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CAT#:0931-T79797-01Size:5 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

2924182-31-8

Target

HIF/HIF Prolyl-Hydroxylase

Related Pathways

Metabolism, Chromatin/Epigenetic

Bioactivity

PHD-IN-1 (compound 80) is a potent PHD2 inhibitor with an IC50 value of ≤5 nM and demonstrates EC50 values of 2.5 μM in EPO Elisa assays in both Caco2-HIF1a-HiBiT-clone-1 and Hep3B cell lines [1].

Smiles

OC=1C2=C(N=C(N3[C@@]4(CN([C@](C3)(C4)[H])C5CC5)[H])C=C2)C=NC1C(NCC=6C=CC(C#N)=NC6)=O

Molecular Formula

C24H23N7O2

Molecular Weight

441.49

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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HY-156526	PHD-IN-1
BA7821-5	PHD-1-IN-1
BA7815-1	HIF-PHD-IN-1
sc-398752	Phd (E-1)
sc-398752 HRP	Phd (E-1) HRP
sc-398752 P	Phd (E-1) P
GTR19013004-01	PHD finger protein 1

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