Anticancer agent 135
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


Anticancer agent 135
Target :
Androgen ReceptorRelated Pathways :
Endocrinology/HormonesBioactivity :
Anticancer agent 135 (compound 26h) is a potent androgen receptor (AR) antagonist that blocks AR nuclear translocation and inhibits AR/AR-V7 heterodimerization to suppress downstream gene transcription, demonstrating strong efficacy in prostate cancer xenograft models [1].Molecular Formula :
C23H21F3N4OSMolecular Weight :
458.5Shipping Conditions :
Cool packStorage Temperature :
-20°C
