BAY 1214784

• Target :

  Others|||GNRH Receptor

• Related Pathways :

  GPCR/G Protein|||Others

• Purity :

  1

• Bioactivity :

  BAY 1214784, a potent, selective, and orally active spiroindoline derivative compound, serves as an antagonist of the human gonadotropin-releasing hormone receptor (hGnRH-R) . It notably reduces plasma luteinizing hormone levels by up to 49%, demonstrating low pharmacokinetic variability and good tolerability. This compound shows promise for research into uterine fibroids.

• Smiles :

  S(=O)(=O)(N1[C@@H](C2(C=3C1=CC=C(C(NCC4=C(Cl)C=C(C(F)(F)F)C=N4)=O)C3)CCS(=O)(=O)CC2)[C@@H]5CC5)C6=CC=C(F)C=C6

• Molecular Formula :

  C29H26ClF4N3O5S2

• Molecular Weight :

  672.11

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1631164-25-4