TAS-108 citrate

CAT: 0931-MF-0144256-01Size: 25 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0144256-01Size:25 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
229634-98-4
Target
Others
Related Pathways
Others
Bioactivity
TAS-108, also known as SR16234, is a synthetic, antiestrogenic steroidal compound with potential antitumor activity. TAS-108 binds to and inhibits estrogenic receptor alpha (ERa), mainly expressed in the mammary gland and uterus and upregulated in estrogen-dependent tumors. Blockage of ERa by TAS-108 prevents the binding and effects of estrogen and may lead to an inhibition of estrogen-dependent cancer cell proliferation. TAS-108 also is a partial agonist of the estrogenic receptor beta (ERb), expressed in many tissues including the central nervous system, urogenital tract, bone and cardiovascular system, thereby exerting a positive effect on these tissues.
Smiles
C(CC(O)=O)(CC(O)=O)(C(O)=O)O.C[C@H]1[C@]2([C@]3([C@@](C)([C@@H](CCOC4=C(OC)C=C(CN(CC)CC)C=C4)CC3)CC[C@@]2(C=5C(C1)=CC(O)=CC5)[H])[H])[H]
Molecular Formula
C39H55NO10
Molecular Weight
697.86
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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