CB2R/FAAH modulator-2

CAT:
931-T67745-01
Size:
1 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
CB2R/FAAH modulator-2 - image 1

CB2R/FAAH modulator-2

  • Target:

    Cannabinoid Receptor|||FAAH
  • Related Pathways:

    GPCR/G Protein|||Metabolism|||Neuroscience
  • Purity:

    0.9952
  • Bioactivity:

    CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting CB2R and FAAH, acting as a CB2R agonist (Ki = 10.8 nM) and FAAH inhibitor (IC50 = 6.2 ?M), with a Ki value of 152.9 nM for CB1R. It has research value in cancer, deleterious inflammatory cascades in neurodegenerative diseases, and COVID-19 infection.
  • Smiles:

    N(C(=O)C1=C(OCC2CCCCC2)C=CC=C1)C34CC5CC(C3)CC(C4)C5
  • Molecular Formula:

    C24H33NO2
  • Molecular Weight:

    367.52
  • Shipping Conditions:

    Cool pack
  • Storage Temperature:

    -20°C
  • CAS Number:

    2876918-68-0