CB2R PAM

CAT: 0931-T37075-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-T37075-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2244579-87-9
Target
Cannabinoid Receptor
Related Pathways
GPCR/G Protein
Purity
0.9909
Bioactivity
CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTP?S binding to CB2 receptors without affecting receptor activity in the absence of agonists. CB2R PAM shows anti-injury activity in a mouse model of neuropathic pain.
Smiles
N(C(=O)C1CCCCCC1)C=2C(=O)N(CC3=CC=C(F)C=C3)C=C(Br)C2C
Molecular Formula
C21H24BrFN2O2
Molecular Weight
435.33
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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