CB2R PAM

• Target:

  Cannabinoid Receptor

• Related Pathways:

  GPCR/G Protein

• Purity:

  0.9909

• Bioactivity:

  CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTP?S binding to CB2 receptors without affecting receptor activity in the absence of agonists. CB2R PAM shows anti-injury activity in a mouse model of neuropathic pain.

• Smiles:

  N(C(=O)C1CCCCCC1)C=2C(=O)N(CC3=CC=C(F)C=C3)C=C(Br)C2C

• Molecular Formula:

  C21H24BrFN2O2

• Molecular Weight:

  435.33

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2244579-87-9