KOR agonist 2

CAT: 0931-MF-0117561-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0117561-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Opioid Receptor
Related Pathways
GPCR/G Protein|||Endocrinology/Hormones|||Neuroscience
Bioactivity
KOR agonist 2 (Compound 23p) is an agonist of the ? opioid receptor (?opioid receptor, KOR) with a Ki of 1.9 nM. In murine models, KOR agonist 2 demonstrates analgesic effects with an ED50 of 1.30 mg/kg. It exhibits high clearance in mice when administered intravenously at 2 mg/kg and shows high metabolism and clearance in liver microsomes.
Molecular Formula
C29H35ClN2O4S
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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