KOR agonist 4

CAT: 0931-T205240-01Size: 10 mgDry Ice: NoHazardous: No

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CAT#:0931-T205240-01Size:10 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Target

Opioid Receptor

Related Pathways

GPCR/G Protein, Neuroscience, Endocrinology/Hormones

Bioactivity

KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.

Molecular Formula

C21H25N3

Molecular Weight

319.44

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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KOR agonist 4

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