Products for Research Use Only

RJG-2051

CAT: 0931-T206799-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T206799-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2851993-77-4
Target
Reductase
Related Pathways
Metabolism, Endocrinology/Hormones
Bioactivity
RJG-2051 is a selective covalent inhibitor of aldo-keto reductase family 1 member C3 (AKR1C3), with an IC50 value of 13 nM. It interferes with the metabolism of substrates such as androgens, estrogens, and prostaglandins through AKR1C3. RJG-2051 holds potential for cancer research.
Smiles
O=C(C1=CC=C(C=C1)S(=O)(=O)N2N=C(N=C2)C3CCCCC3)N4CCN(C=5C=CC=CC5OC)CC4
Molecular Formula
C26H31N5O4S
Molecular Weight
509.62
Shipping Conditions
Ice Packs
Storage Temperature
-20°C