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Anticancer agent 258

CAT: 0931-T203128-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T203128-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2891984-12-4
Target
Others, Orphan Receptor
Related Pathways
Others, GPCR/G Protein
Bioactivity
Anticanceragent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates nuclear receptor activity. It exhibits an EC50 of 63 nM for Nurr in N2A cells and an IC50 of 0.1 pM for Nur77 in HEK293 cells. Anticanceragent 258 is applicable in studies related to cancer, metabolic disorders, and neurological diseases.
Smiles
FC=1C=CC(=CC1)C=2N=C3N(N2)C=C(C=4C=CC=C(F)C4)N3C
Molecular Formula
C17H12F2N4
Molecular Weight
310.3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C