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PAR4 antagonist 8

CAT: 0931-T201684-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T201684-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
MDM-2/p53, Protease-activated Receptor
Related Pathways
GPCR/G Protein, Apoptosis
Bioactivity
PAR4 antagonist8 (Compound 20f) is an effective oral and selective PAR4 antagonist with an IC50 of 15.32 nM, boasting favorable pharmacokinetic properties. It effectively inhibits human platelet aggregation induced by PAR4 agonists (IC50=6.39 nM) and also suppresses platelet aggregation in mice. PAR4 antagonist8 is utilized in anti-thrombotic research.
Molecular Formula
C28H19F2N5O4S
Molecular Weight
559.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C