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PROTAC EZH2 Degrader-3

CAT: 0931-T200955-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T200955-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Histone Methyltransferase, PROTACs, Apoptosis
Related Pathways
Apoptosis, PROTAC, Chromatin/Epigenetic
Bioactivity
PROTAC EZH2 Degrader-3 (compound ZJ-20) is a potent EZH2 degrader that exhibits strong inhibitory effects not only on EZH2 protein expression but also on the levels of other PRC2 subunits and H3k27me3 protein. Additionally, PROTAC EZH2 Degrader-3 demonstrates antiproliferative activity by blocking the cell cycle at the G0-G1 phase and inducing apoptosis (cell death) . At a concentration of 5 μM and over a period of 24 hours, it effectively suppresses the expression of these critical proteins involved in cell regulation and growth.
Smiles
O=C1NC(=O)C=2C1=C3C4=CC(=CC=C4NC3=C5C2CCC5)C(=O)CCC(=O)O
Molecular Formula
C56H68N8O8
Molecular Weight
981.19
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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