HDAC-IN-57

• Description:

  HDAC-IN-57 is an orally active pan-inhibitor of histone deacetylase (HDAC), inhibiting HDAC1, HDAC2, HDAC6, and HDAC8 with IC50 values of 2.07 nM, 4.71 nM, 2.4 nM, and 107 nM, respectively. HDAC-IN-57 inhibits LSD1 with an IC50 value of 1.34 μΜ. HDAC-IN-57 has anti-tumor activity and can induce apoptosis.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  377.39

• Molecular Formula:

  C21H19N3O4

• Notes:

  Research use only, not for human use.

• Receptor:

  HDAC | Apoptosis

• CAS Number:

  2716217-79-5