HS-276

• Description:

  HS-276 is a highly selective, orally active inhibitor of TAK1 (Ki: 2.5 nM) . HS-276 significantly inhibits TAK1 (IC50: 8.25 nM), CLK2 (IC50: 29 nM), GCK (IC50: 22 nM), ULK2 (IC50: 63 nM), MAP4K5 (IC50. HS-276 can be used to study rheumatoid arthritis (RA) .

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  419.52

• Molecular Formula:

  C24H29N5O2

• Notes:

  Research use only, not for human use.

• Receptor:

  MAPK

• CAS Number:

  2767422-72-8