HS 014

• Description:

  Potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively) . Increases food intake in rats and nociception in mice following central administration in vivo. Also inhibits IL-1β-induced Fos expression in the paraventricular hypothalamus.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  1563.77

• Molecular Formula:

  C71H94N20O17S2

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  207678-81-7