HS 024

• Description :

  Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively) . Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  1266.5

• Molecular Formula :

  C58H79N19O10S2

• Notes :

  Research use only, not for human use.

• Receptor :

  ——

• CAS Number :

  212370-59-7