HS 024

• Description:

  Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively) . Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  1266.5

• Molecular Formula:

  C58H79N19O10S2

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  212370-59-7