Products for Research Use Only

GSK-5959

CAT: 0421-82066Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0421-82066Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GSK-5959 exhibits >100-fold selectivity for BRPF1 (IC50= 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.
CAS Number
901245-65-6
Format
Solid
Molecular Formula
C22H26N4O3
Shipping Conditions
Room Temperature
Storage Conditions
At least 6 months at -20°C.
Calculated Molecular Weight
394.5 Da