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GSK-5959

CAT: 0026-B2343-5Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0026-B2343-5Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GSK-5959 is a potent and selective BRPF1 (BR140 or Peregrin) bromodomain inhibitor (IC₅₀ = 80 nM). GSK-5959 displays >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains. BRPF1 (bromodomain and PHD finger containing protein 1) is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.
Shipping Conditions
Gel Pack
Storage Conditions
-20ºC
Shelf Life
36 months