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GLPG0974

CAT: 0804-HY-12940-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-12940-01Size:5 mg
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Description
GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM.
CAS Number
[1391076-61-1]
UNSPSC
12352005
Target
Free Fatty Acid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/GLPG0974.html
Purity
98.12
Solubility
DMSO : 200 mg/mL (ultrasonic)
Smiles
O=C(O)CCCN(C([C@]1(C)N(C(C2=CSC3=CC=CC=C32)=O)CC1)=O)CC4=CC=CC(Cl)=C4
Molecular Formula
C25H25ClN2O4S
Molecular Weight
485.00
References & Citations
[1]Pizzonero M, et al. Discovery and optimization of an azetidine chemical series as a free fatty acid receptor 2 (FFA2) antagonist: from hit to clinic. J Med Chem. 2014 Dec 11;57 (23) :10044-57.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 2

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T15388-01GLPG0974
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A21466-1GLPG0974 1mg
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