Products for Research Use Only

CAF-382

CAT: 0013-GTR19230408-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19230408-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CAF-382 (compound B1) is a SNS-032 analog functioning as a potent CDKL5 and pan-CDK inhibitor, with additional modest activity against GSK3α/β (IC50 >1.8 μM) . It blocks CDKL5-mediated E2 domain phosphorylation and is a valuable chemical probe for studying kinase signaling in neurological disease models, both in vitro and in vivo.
Field of Research
Cell Biology, Signal Transduction
Molecular Formula
C16H22N4O2S2
Molecular Weight
366.5
Storage Conditions
-20°C
Notes
For research use only.