Products for Research Use Only

BMS-819881

CAT: 0013-GTR19203906-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19203906-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
BMS-819881 is a potent and selective antagonist of the melanin-concentrating hormone receptor 1 (MCHR1), exhibiting a Ki of 7 nM for the rat receptor. It also acts as a CYP3A4 inducer with an EC50 of 13 μM. This small molecule is a valuable research tool for studying energy homeostasis, sleep regulation, and metabolic disorders in both in vitro and in vivo models.
CAS Number
1197420-05-5
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
O=C1C2=C (C=C (S2) C3=CC=C (Cl) C=C3) N=CN1C4=CC (OC) =C (OC[C@H] (O) C5CC5) C=C4
Molecular Formula
C24H21ClN2O4S
Molecular Weight
468.95
Storage Conditions
-20°C
Notes
For research use only.