BMS-819881

• Target :

  Cytochromes P450|||Melanin-concentrating Hormone Receptor (MCHR) |||GPCR

• Related Pathways :

  GPCR/G Protein|||Endocrinology/Hormones|||Metabolism

• Bioactivity :

  BMS-819881, a melanin-concentrating hormone receptor 1 (MCHR1) antagonist, binds rat MCHR1 with a Ki of 7 nM, and is selective and potent for CYP3A4 activity with an EC50 of 13 ?M.

• Smiles :

  O=C1C2=C(C=C(S2)C3=CC=C(Cl)C=C3)N=CN1C4=CC(OC)=C(OC[C@H](O)C5CC5)C=C4

• Molecular Formula :

  C24H21ClN2O4S

• Molecular Weight :

  468.95

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1197420-05-5