BMS-819881

• Target:

  Cytochromes P450|||Melanin-concentrating Hormone Receptor (MCHR) |||GPCR

• Related Pathways:

  GPCR/G Protein|||Endocrinology/Hormones|||Metabolism

• Bioactivity:

  BMS-819881, a melanin-concentrating hormone receptor 1 (MCHR1) antagonist, binds rat MCHR1 with a Ki of 7 nM, and is selective and potent for CYP3A4 activity with an EC50 of 13 ?M.

• Smiles:

  O=C1C2=C(C=C(S2)C3=CC=C(Cl)C=C3)N=CN1C4=CC(OC)=C(OC[C@H](O)C5CC5)C=C4

• Molecular Formula:

  C24H21ClN2O4S

• Molecular Weight:

  468.95

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1197420-05-5