Products for Research Use Only

EST73502 hydrochloride

CAT: 0013-GTR19184479-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19184479-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
EST73502 hydrochloride is an orally bioavailable, brain-penetrant small molecule functioning as a dual μ-opioid receptor agonist (Ki=64 nM) and σ1 receptor antagonist (Ki=118 nM) . It demonstrates analgesic efficacy in preclinical models while showing a potentially improved side-effect profile, making it a candidate for neuropathic pain and addiction research.
CAS Number
2307458-82-6
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Smiles
CCN1CC2 (CCN (CCC3=CC (F) =CC=C3F) CC2) O[C@H] (C) C1=O
Molecular Formula
C19H27ClF2N2O2
Molecular Weight
388.88
Storage Conditions
-20°C
Notes
For research use only.