Products for Research Use Only

Mirogabalin (Standard)

CAT: 0804-HY-12650R-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-12650R-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Mirogabalin (Standard) is the analytical standard of Mirogabalin. This product is intended for research and analytical applications. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS.
CAS Number
1138245-13-2
Product Name Alternative
DS5565 (Standard)
UNSPSC
12352211
Target
Calcium Channel; Reference Standards
Type
Reference Standards
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling; Others
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/mirogabalin-standard.html
Smiles
O=C(O)C[C@]1(CN)[C@]2([H])C=C(CC)C[C@]2([H])C1
Molecular Formula
C12H19NO2
Molecular Weight
209.28
References & Citations
[1]Vinik A, et al. Efficacy and safety of Mirogabalin (DS-5565) for the treatment of diabetic peripheral neuropathic pain: a randomized, double-blind, placebo- and active comparator-controlled, adaptive proof-of-concept phase 2 study. Diabetes Care. 2014 Dec|[2]Hutmacher MM, et al. Exposure-response modeling of average daily pain score, and dizziness and somnolence, forMirogabalin (DS-5565) in patients with diabetic peripheral neuropathic pain. J Clin Pharmacol. 2016 Jan;56 (1) :67-77.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards