Mirogabalin-13C2,d1 (Mixture of Diastereomers)

• UNSPSC Description:

  Mirogabalin-13C2,d1 (Mixture of Diastereomers) is a C13 and deuterium labeled Mirogabalin. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS[1].

• Target Antigen:

  Isotope-Labeled Compounds

• Type:

  Isotope-Labeled Compounds

• Related Pathways:

  Others

• Field of Research:

  Others

• Solubility:

  10 mM in DMSO

• Smiles:

  O=[13C](O)[13CH2]C1(C([2H])([H])N)[C@]2([H])C=C(CC)C[C@]2([H])C1

• Molecular Weight:

  212.28

• References & Citations:

  [1]Vinik A, et al. Efficacy and safety of Mirogabalin (DS-5565) for the treatment of diabetic peripheral neuropathic pain: a randomized, double-blind, placebo- and active comparator-controlled, adaptive proof-of-concept phase 2 study. Diabetes Care. 2014 Dec^[1].

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported