Mirogabalin-13C2,d1 (Mixture of Diastereomers)

Mirogabalin-13C2,d1 (Mixture of Diastereomers)

• UNSPSC Description: Mirogabalin-13C2,d1 (Mixture of Diastereomers) is a C13 and deuterium labeled Mirogabalin. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS[1].
• Target Antigen: Isotope-Labeled Compounds
• Type: Isotope-Labeled Compounds
• Related Pathways: Others
• Field of Research: Others
• Solubility: 10 mM in DMSO
• Smiles: O=[13C](O)[13CH2]C1(C([2H])([H])N)[C@]2([H])C=C(CC)C[C@]2([H])C1
• Molecular Weight: 212.28
• References & Citations: [1]Vinik A, et al. Efficacy and safety of Mirogabalin (DS-5565) for the treatment of diabetic peripheral neuropathic pain: a randomized, double-blind, placebo- and active comparator-controlled, adaptive proof-of-concept phase 2 study. Diabetes Care. 2014 Dec^[1].
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported