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Gabapentin enacarbil

CAT: 0804-HY-16216-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-16216-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Gabapentin enacarbil (XP-13512) is a prodrug of Gabapentin designed to be absorbed throughout the intestine by high-capacity nutrient transporters. Gabapentin is a potent, orally active P/Q type Ca2+ channel blocker. Gabapentin enacarbil can be used for the study of Restless Legs Syndrome (RLS) and postherpetic neuralgia (PHN)[2].
CAS Number
478296-72-9
Product Name Alternative
XP-13512
UNSPSC
12352211
Hazard Statement
H302, H315, H319, H335
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Gabapentin-enacarbil.html
Concentration
10mM
Purity
98.0
Solubility
DMSO : ≥ 100 mg/mL|Ethanol : 100 mg/mL (ultrasonic)
Smiles
O=C(O)CC1(CNC(OC(OC(C(C)C)=O)C)=O)CCCCC1
Molecular Formula
C16H27NO6
Molecular Weight
329.39
Precautions
H302, H315, H319, H335
References & Citations
[1]Cundy KC, et al. XP13512 [ (+/-) -1- ([ (alpha-isobutanoyloxyethoxy) carbonyl] aminomethyl) -1-cyclohexane acetic acid], a novel gabapentin prodrug: I. Design, synthesis, enzymatic conversion to gabapentin, and transport by intestinal solute transporters. J Pharmacol Exp Ther. 2004 Oct;311 (1) :315-23.|[2]Cundy KC, et al. XP13512 [ (+/-) -1- ([ (alpha-isobutanoyloxyethoxy) carbonyl] aminomethyl) -1-cyclohexane acetic acid], a novel gabapentin prodrug: II. Improved oral bioavailability, dose proportionality, and colonic absorption compared with gabapentin in rats and monkeys. J Pharmacol Exp Ther. 2004 Oct;311 (1) :324-33.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, protect from light, stored under nitrogen)
Scientific Category
Reference compound1
Clinical Information
Launched

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