BigLEN (rat)

• Target:

  GPCR

• Related Pathways:

  Endocrinology/Hormones|||GPCR/G Protein

• Bioactivity:

  Potent GPR171 agonist (EC50 = 1.6 nM) . ProSAAS-derived peptide. Regulates body weight in mice and promotes the outgrowth of neurites in Neuro2A cells.

• Smiles:

  C (=O) ([C@H]1N (C ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC (=O) [C@H]2N (C ([C@@H] (NC ([C@@H] (NC (=O) [C@H]3N (C ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@H] (CC (C) C) N) =O) CCC (O) =O) =O) CC (N) =O) =O) CO) =O) CO) =O) CCC3) CCC (N) =O) =O) C) =O) CCC2) C) =O) CCCNC (=N) N) =O) CCCNC (=N) N) =O) CC (C) C) =O) CC (C) C) =O) CCC1) N4[C@H] (C (O) =O) CCC4

• Molecular Formula:

  C76H128N24O23

• Molecular Weight:

  1746

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  369377-66-2