PG 106 acetate

• Target :

  Melanocortin Receptor

• Related Pathways :

  GPCR/G Protein|||Neuroscience

• Purity :

  0.9824

• Bioactivity :

  PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.

• Smiles :

  CCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCC/N=C(N)\N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O

• Molecular Formula :

  C53H73N13O11

• Molecular Weight :

  1068.23

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C