EPI-7170

• Target :

  Others|||Androgen Receptor

• Related Pathways :

  Others|||Endocrinology/Hormones

• Bioactivity :

  EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs) . EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC) .

• Smiles :

  C(C)(C)(C1=CC(Cl)=C(OC[C@@H](CCl)O)C(Cl)=C1)C2=CC=C(OC[C@@H](CNS(C)(=O)=O)O)C=C2

• Molecular Formula :

  C22H28Cl3NO6S

• Molecular Weight :

  540.88

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2139288-26-7