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UNC0379 TFA

CAT: 0931-T63705-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0931-T63705-01Size:100 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1620401-83-3
Target
Others, Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
UNC0379 TFA is a selective, substrate-competitive inhibitor of lysine methyltransferase SETD8 (KMT5A) with an IC50 of 7.3 μM, and demonstrates good selectivity for 15 other methyltransferases.
Smiles
OC(=O)C(F)(F)F.COc1cc2nc(nc(NCCCCCN3CCCC3)c2cc1OC)N1CCCC1
Molecular Formula
C25H36F3N5O4
Molecular Weight
527.589
Shipping Conditions
Ice Packs
Storage Temperature
-20°C