UNC0379 TFA

• Target:

  Others|||Histone Methyltransferase

• Related Pathways:

  Chromatin/Epigenetic|||Others

• Bioactivity:

  UNC0379 TFA is a selective, substrate-competitive inhibitor of lysine methyltransferase SETD8 (KMT5A) with an IC50 of 7.3 ?M, and demonstrates good selectivity for 15 other methyltransferases.

• Smiles:

  OC(=O)C(F)(F)F.COc1cc2nc(nc(NCCCCCN3CCCC3)c2cc1OC)N1CCCC1

• Molecular Formula:

  C25H36F3N5O4

• Molecular Weight:

  527.589

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1620401-83-3