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GABAA receptor agent 5

CAT: 0931-T61668-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T61668-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1808389-92-5
Target
GABA Receptor
Related Pathways
Membrane transporter/Ion channel, Neuroscience
Purity
0.9939
Bioactivity
GABAA receptor agent 5 demonstrates antagonist activity across multiple GABAA receptor subtypes, and GABAA receptor agent 5 exhibits IC50 values of 0.24, 0.088, 0.068, 0.33, 0.79, 0.32, 0.079, and 0.051 μM for α1β2δ, α4β1δ, α4β2δ, α6β2δ, α1β2γ2, α2β2γ2, α3β2γ2, and α5β2γ2 receptor configurations, respectively. GABAA receptor agent 5 (compound 018) thereby provides a precise pharmacological tool for characterizing subtype-selective GABAA receptor inhibition and supports mechanistic neuropharmacology studies focused on inhibitory synaptic signaling and therapeutic antagonist development.
Smiles
O=C(NC1=CC=CC(=C1)C(=O)N2CCC3(CCNCC3)CC2)C=4SC=CC4
Molecular Formula
C21H25N3O2S
Molecular Weight
383.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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