ARN-3236

• Target:

  AMPK|||SIK

• Related Pathways:

  Chromatin/Epigenetic|||PI3K/Akt/mTOR signaling

• Purity:

  0.997

• Bioactivity:

  ARN-3236 is an orally active and selective inhibitor of salt-inducible kinase 2 (SIK2), with IC50 values of <1 nM for SIK2, 21.63 nM for SIK1, and 6.63 nM for SIK3. ARN-3236 exhibits anti-cancer activity.

• Smiles:

  COc1ccc(-c2c[nH]c3nccc(-c4ccsc4)c23)c(OC)c1

• Molecular Formula:

  C19H16N2O2S

• Molecular Weight:

  336.41

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1613710-01-2