Products for Research Use Only

ML-030

CAT: 0931-T5496-01Size: 1 mL - 10 mM (in DMSO)Dry Ice: NoHazardous: No
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CAT#:0931-T5496-01Size:1 mL - 10 mM (in DMSO)
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1013750-77-0
Target
PDE
Related Pathways
Metabolism
Purity
0.9824
Bioactivity
ML-030 is a potent and selective inhibitor of PDE4 (PDE4A, PDE4A1, PDE4B1, PDE4B2, PDE4C1, and PDE4D2 with IC50 of 6.7 nM, 12.9 nM, 48.2 nM, 37.2 nM, 452 nM and 49.2 nM, respectively)
Smiles
COc1ccc(OC)c(c1)-c1nnc2SCC(=Nn12)c1ccc(OC)c(OC)c1
Molecular Formula
C20H20N4O4S
Molecular Weight
412.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C