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PDE12-IN-1

CAT: 0931-T39796-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T39796-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2259620-80-7
Target
Others, PDE
Related Pathways
Metabolism, Others
Bioactivity
PDE12-IN-1 is a powerful and specific inhibitor of PDE12, exhibiting a pIC 50 value of 9.1 for enzyme inhibition. It effectively enhances levels of 2′,5′-linked adenylate polymers (2-5A), with a pEC 50 value of 7.7. Additionally, PDE12-IN-1 demonstrates antiviral activity.
Smiles
CCn1cc(-c2nc3cc(Br)c(cc3n2C)C(=O)N2CCO[C@@H]([C@H]2CO)c2ccc(F)cc2)c2ccc(cc12)C#N
Molecular Formula
C31H27BrFN5O3
Molecular Weight
616.491
Shipping Conditions
Ice Packs
Storage Temperature
-20°C