VGSC blocker-1

• Target:

  Others|||Sodium Channel

• Related Pathways:

  Others|||Membrane transporter/Ion channel

• Bioactivity:

  VGSC blocker-1 is a powerful small molecule that serves as a blocker for the neonatal isoform of the VGSC subtype known as Nav1.5 (nNav1.5) . It effectively blocks INa peak currents by 34.9% at a concentration of 1 ?M, and demonstrates a 0.3% inhibition of cell invasion at the same concentration in the MDA-MB-231 human breast cancer cell line, without compromising cell viability.

• Smiles:

  Fc1ccc(cc1)C(CCCNCCCN1CCCCC1)c1ccc(F)cc1

• Molecular Formula:

  C24H32F2N2

• Molecular Weight:

  386.52

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2230472-55-4