TRPV2-selective blocker 1

CAT: 0931-T80930-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0931-T80930-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2242724-49-6
Target
TRP/TRPV Channel|||Others
Related Pathways
Others|||Membrane transporter/Ion channel
Bioactivity
TRPV2-selective blocker 1 (compound IV2-1) is a selective inhibitor of the TRPV2 channel, with an IC50 value of 6.3 ?M, specifically targeting the TRPV2 channel without affecting TRPV1, TRPV3, or TRPV4 channels, and effectively suppresses TRPV2-mediated calcium influx in macrophages, inhibiting their phagocytic activity [1].
Smiles
O=C(C)CC(C(=C1SCCS1)C=2C=CC=CC2)C
Molecular Formula
C15H18OS2
Molecular Weight
278.43
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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