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CAY10573

CAT: 0931-T37829-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T37829-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
853652-40-1
Target
PPAR, Others
Related Pathways
Others, DNA Damage/DNA Repair, Metabolism
Bioactivity
The peroxisome proliferator-activated receptors (PPARs) are lipid-activated transcription factors often used as drug targets for the treatment of metabolic disorders. CAY10573 is a PPAR agonist that displays potent binding at PPARα, γ, and δ with IC50 values of 113, 50, and 223 nM, respectively. It potently transactivates PPARα, γ, and δ with EC50 values of 8, 70, and 500 nM, respectively. CAY10573 demonstrates stronger binding and functional activity for PPARγ than the antidiabetic compound rosiglitazone (IC50 = 92 nM; EC50 = 220 nM) .
Smiles
C(CC)C=1C2=C(C=C(C(=O)C3=CC=CC=C3)C=C2)C=CC1OCCCOC=4C=C5C(=CC4)N(CC(O)=O)C=C5
Molecular Formula
C33H31NO5
Molecular Weight
521.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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MBS5798633CAY10573

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