TP-238

• Target:

  Others|||Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic|||Others

• Bioactivity:

  TP-238, a potent and selective dual CECR2/BPTF probe, exhibits IC50 values of 30 nM and 350 nM, respectively. Additionally, it inhibits BRD9 with a pIC50 of 5.9, demonstrating lesser activity against another 338 kinases [1] [2].

• Smiles:

  N(CCCN1C=CC=N1)C2=CC(=NC(S(C)(=O)=O)=N2)C3=CC=C(OCCCN(C)C)C=C3

• Molecular Formula:

  C22H30N6O3S

• Molecular Weight:

  458.58

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2415263-04-4