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AVN-101

CAT: 0931-T26690-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-T26690-01Size:1 mg
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AVAILABILITY
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1061354-48-0
Target
Histamine Receptor|||5-HT Receptor|||Adrenergic Receptor
Related Pathways
Immunology/Inflammation|||GPCR/G Protein|||Neuroscience
Purity
0.9973
Bioactivity
AVN-101 is a highly potent 5-HT7 receptor antagonist with a Ki value of 153 pM. AVN-101 also exhibits considerable affinity for histamine H1 (Ki value of 0.58 nM) and adrenergic ?2A, ?2B and ?2C (Ki values ??of 0.41-3.6 nM) receptors. AVN-101 has shown good oral bioavailability and brain-blood barrier permeability, low toxicity and reasonable efficacy in animal models of central nervous system diseases.
Smiles
Cl.CN1CCC2=C(C1)C1=CC(C)=CC=C1N2CCC1=CC=CC=C1
Molecular Formula
C21H25ClN2
Molecular Weight
340.89
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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