GSK-5959

• CAS Number :

  901245-65-6

• Target :

  Epigenetic Reader Domain

• Related Pathways :

  Chromatin/Epigenetic

• Purity :

  0.9877

• Bioactivity :

  GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM) . The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.

• Smiles :

  COc1ccccc1C(=O)Nc1cc2n(C)c(=O)n(C)c2cc1N1CCCCC1

• Molecular Formula :

  C22H26N4O3

• Molecular Weight :

  394.47

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C