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PD153035 hydrochloride

CAT: 0931-T1761-01Size: 1 mL - 10 mM (in DMSO)Dry Ice: NoHazardous: No
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CAT#:0931-T1761-01Size:1 mL - 10 mM (in DMSO)
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
183322-45-4
Target
EGFR
Related Pathways
Angiogenesis, JAK/STAT signaling, Tyrosine Kinase/Adaptors
Purity
>99.99%
Bioactivity
PD153035 hydrochloride (ZM 252868) is a effective and selective inhibitor of EGFR (Ki: 5.2 pM, IC50: 29 pM) ; few influence against FGFR, PGDFR, InsR, CSF-1, and Src.
Smiles
Cl.COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OC
Molecular Formula
C16H15BrClN3O2
Molecular Weight
396.67
Shipping Conditions
Ice Packs
Storage Temperature
-20°C